平安! 发表于 2011-11-9 19:57 R0 q( j3 _2 w+ R3 S: X
Pazopanib (100 mg/kg/day free base equivalent)
3 e" ~# V6 v0 ~6 I" R$ q 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。0 G$ g' Z% g: O7 s" H* s+ {
搜索了一下,原料一大堆。5 x; H2 G. @4 O, s3 a$ }
. D, |1 r/ w6 H u' m; g对不起!100mg/kg是用于移植瘤的,我弄错了。
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4 t8 X8 L ~5 b; j6 \以下是正版说明书的推荐用量。2 x( O$ k, @& K
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--------------------- DOSAGE AND ADMINISTRATION ----------------6 {6 }+ A) G0 ^
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) # V3 h5 ]+ N) t7 b
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 9 p+ X& W5 N8 A4 {
---------------------DOSAGE FORMS AND STRENGTHS --------------4 u9 `7 o2 W" G( X
200 mg tablets. (3)
+ A6 l& A7 c& z/ \-------------------------------CONTRAINDICATIONS------------------------ |